Back to Peptides

DSIP (Delta Sleep-Inducing Peptide)

Neuroprotective & Cognitive Enhancers

DSIP (Delta Sleep-Inducing Peptide) is a short neuropeptide with documented ability to promote deep sleep, reduce stress, and modulate circadian rhythms. Often used to support recovery, anxiety reduction, and HPA balance, DSIP has broad experimental interest for its neuroendocrine effects.

Reconstitute
3 mL BAC + 5mg vial
17 mcg/unit
Daily Range
100–400 mcg Subcutaneous (SQ)
30–60 minutes before bedtime
Standard Dose
200 mcg
Cycle
4–8 weeks
then reassess
DSIPdelta sleep peptidesleep optimizationanxiolytic peptideHPA regulation

Dosing & Reconstitution Guide

In rodent studies, DSIP was used at 100–500 μg/kg IP or IV. Human effects are not well characterized. Not approved for sleep therapy or clinical use.

Standard / Gradual Approach

5mg Vialstandard
PhaseDoseVolume
Week 1100 mcg6 units (0.06 mL)
Week 2150 mcg9 units (0.09 mL)
Week 3200 mcg12 units (0.12 mL)
Weeks 4–8250–300 mcg15–18 units (0.15–0.18 mL)

Standard / Gradual Approach

5mg Vialadvanced
PhaseDoseVolume
Week 5350–400 mcg21–24 units (0.21–0.24 mL)
Weeks 6–8+400–500 mcg24–30 units (0.24–0.30 mL)

Standard / Gradual Approach

10mg Vialstandard
PhaseDoseVolume
Week 1100 mcg3 units (0.03 mL)
Week 2150 mcg5 units (0.05 mL)
Week 3200 mcg6 units (0.06 mL)
Weeks 4–8250–300 mcg8–9 units (0.08–0.09 mL)

Protocol Summary

Subcutaneous (SQ): 30–60 minutes before bedtime · Dose range 100400 mcg with gradual titration
Cycle Length: 4–8 weeks typical; reassess before extending

Frequency & Cycling

SubQ Injection

Use nightly for 2–4 weeks, then cycle off for 1–2 weeks to prevent receptor fatigue. Take 30–60 minutes before bed.

🧪 Quick Start

Vial Size
5 mg
BAC Water
3 mL
Concentration
1.67 mcg/unit
Starting Dose
100 mcg before bedtime
Maintenance Dose
100 mcg nightly

Potential Benefits & Use Cases

DSIP is a research-use-only peptide. It is not approved for sleep support or therapeutic use in any country.
Promotes deeper, more restorative slow-wave sleep and improves subjective sleep quality (limited human data)
Demonstrates stress-protective and anxiolytic-like effects (preclinical)
Does not appear to induce pharmacological tolerance with continued use (limited human data)
Supports immune cell proliferation and tumor growth reduction in animal models (preclinical)
Clinical data Strong preclinical Limited data

Mechanism of Action

Modulates delta sleep EEG activity via hypothalamic pathways
Inhibits corticotropin-releasing hormone (CRH), reducing stress
Stabilizes neuronal excitability and acts as a mild neuropeptide anxiolytic
May influence melatonin, serotonin, and other neuroendocrine rhythms

Lifestyle & Optimization

timing

Administer at bedtime for sleep induction.

diet

Limit stimulants (caffeine) before bed.

exercise

Regular exercise earlier in the day — not close to bedtime.

sleep

Consistent sleep-wake schedules. Cool, dark, quiet environment. Limit blue light before bed. Stress management.

Side Effects & Safety

Common Side Effects

Morning fatigue/lethargy if dose too high or wrong timing
Headache, dizziness, nausea
Stomach pain/GI issues

Contraindications & Warnings

May interact with GABA/NMDA receptor activity; risk with sedatives and alcohol

Long-Term Safety Data

Long-term safety not established; not FDA-approved

🧮 Dose Calculator

Concentration
16.7
mcg/unit
Draw Volume
30
units (0.300 mL)
For a 500 mcg dose, draw 30 units on a U-100 insulin syringe
🧬

Bioavailability & Absorption

SubQ Injection
High absorption and CNS penetration observed in animal models
Oral Administration
Not viable due to rapid degradation
Half-Life
15–30 minutes systemically; longer CNS effect suspected
Degradation
Primarily metabolized by peptidases and hepatic clearance
Tissue Specificity
Acts on hypothalamus, pineal gland, hippocampus, and reticular formation
⚗️

Peptide Details

Molecular Weight
848.8
Formula
C35H48N10O15
Sequence
Trp-Ala-Gly-Gly-Asp-Ala-Ser-Gly-Glu
⚖️

Legal Status & Regulatory

RegionStatus
FDANot Approved
EUNot Approved
AustraliaNot Approved
CanadaNot Approved

Storage Instructions

Lyophilized (Powder)
Store lyophilized powder at -20°C for long-term or 2-8°C for up to 6 months. Protect from light and moisture. Do not freeze reconstituted solution. Avoid repeated temperature fluctuations.
Reconstituted (Mixed)
Refrigerate at 2-8°C. Use within 3-4 weeks.